Pharmaceutical Raw Materials Fladrafinil / CRL-40,941 CAS 90212-80-9 For Intelligence Development

CAS: 90212-80-9

MF: C15H13F2NO3S

MW: 325.3304264

Synonyms: AcetaMide, 2-[[bis(4-fluorophenyl)Methyl]sulfinyl]-N-hydroxy-;2-[bis(4-fluorophenyl)Methyl]sulfinylethanehydroxaMic acid;Fladrafinil;Fladrafinil (Bisfluoroadrafinil);2-[[Bis(4-fluorophenyl)methyl]sulfinyl]-N-hydroxyacetamide;CRL-40,941;Fladrafinil, Bisfluroadrafinil

What is Fladrafinil

Fladrafinil is also referred to as CRL-40,941 or fluorafinil. It is a wakefulness-promoting agent that is found in the eugeroic classification of drugs. Fladrafinil is closely related to adrafinilandmodafinil. Though it's chemical composition and effects are very similar, it is capable of producing anti-aggressive effects while adrafinildoesn't have this ability. Fladrafinil is the bis(p-fluoro) ring-substituted derivative ofadrafinil. It promotes wakefulness and thought acceleration. It increases cognitive function, motivation, and improves memory as it works on dopamine and histamine neurotransmitters in the brain.

Effects

The drug is reported to have little or no side effects when taken at the correct dose over a short period of time. Fladrafinil is ONLY designed and intended for short term use. Long-term use and misuse of the drug can affect our brain in many ways. This medicine blocks the reuptake of dopamine and norepinephrine in the presynaptic cleft immediately upon being released. Long-term use of the drug causes lesions on cerebral blood pathways and brain injury affects the efficiency of neurotransmitter substances in our brain.
 

Dosage

Fladrafinil is 3-4 more potent thanadrafinil. New users should start with 30-80 mgs within 14-16 hours daily, and anadrafinil moderate dose is between 30-100 mg per day. The dosage to be increased as the effects are being experienced as the body reacts towards the dose. Dosage should not exceed 200mgs per day.

Fladrafinil causes the following in human body

1) Improves memory as it works on dopamine and histamine that are neurotransmitter in the brain

2) Increases cognitive function since it boosts the working capacity of the brain when one is in an awkward situation.

3) It's used to treat insomnia and depression.

4) It promotes consciousness

5) It increases motivation, making one to do a lot of activities without exhaustion.

How to use

Fladrafinil is slightly soluble in water. The drug can be taken in the form of capsule or tablet, the drug is taken orally with or without food. It's highly recommended for the drug to be taken early in the morning so that one will experience the impacts of the drug throughout the day. Prior to start work, it will work well if you take 1 hour before you start your intended duty.

Long-term use

- Insomnia cases can be experienced, since it affects the sleeping pattern, it will be difficult to regain the normal sleeping cycle over short period after leaving the drug
- Brain damage and injury can occur as the drug influence the action of neurotransmitter substances in the synapse by blocking them.

 

Short-term use

The drug is reported to have little or no effects when taken at the correct dose. The most common effect on short-term use is just like the ects of other drugs in the nootropic products. These are;
- It causes a headache as it's associated with dehydration
- Increases blood pressure due to vasoconstriction of blood vessels
- Stomach discomfort due to poor digestion
- Aggression and
- Confusion.
 

Nootropic- Brain Health

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