Place of Origin: | CHINA |
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Brand Name: | TINGYI |
Certification: | GMP , ISO 9001:2008 |
Model Number: | 81409-90-7 |
Minimum Order Quantity: | 1g powder or 1 vial (10mg) |
Price: | 1g powder : 3380 USD ; 1 vial (10mg) : 90 USD |
Packaging Details: | Stealth And Discreet Packaging |
Delivery Time: | Within 7 Working Days |
Payment Terms: | Bank Transfer - Bitcoin - Western Union - MoneyGram |
Supply Ability: | 10 G/Month |
Product Name: | Cabergoline | Other Name: | Dostinex ; Caber |
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CAS: | 81409-90-7 | MF: | C26H37N5O2 |
MW: | 451.6 | Specification: | 10mg/vial |
High Light: | anti estrogen products,anti estrogen drugs |
Cabergoline
Basic Details :
Product Name: Cabergoline
Synonyms: Dostinex ; Caber
CAS: 81409-90-7
MF: C26H37N5O2
MW: 451.6
EINECS: 200-419-0
Melting point 102-104°C
storage temp. Store at +4°C
solubility DMSO: ≥10mg/mL
Description:
Cabergoline is a dopamine receptor agonist. It works by reducing the amount of prolactin (a hormone) that is released from the pituitary gland. Cabergoline is used to treat a hormone imbalance in which there is too much prolactin in the blood (also called hyperprolactinemia).
Cabergoline is a dopamine agonist. Dopamine is a chemical, found in the brain, which transmits nerve impulses and is involved in the formation of epinephrine. More likely than not, this is why the Life-Extentionistas are very big on this drug. Dopamine is also released by the hypothalamus, and hormone can inhibit the release of prolactin from the anterior lobe of the pituitary, so given all the bad things that we have already seen to be a result of excess
Application:
Cabergoline is used to treat high levels of prolactin hormone in your body. High levels of prolactin in women can cause symptoms such as unwanted breast milk and missed periods and can cause difficulty becoming pregnant. High levels of prolactin in men can cause symptoms such as enlarged breasts and decreased sexual ability/desire. Cabergoline is an ergot medication and works by blocking the release of prolactin from the pituitary gland.
Cabergoline will help you reduce the chance of any of these prolactin related side-effects. It has actually been shown in numerous studies to have a very high success rate in lowering prolactin and prolactin related conditions and side-effects. In fact, for management of hyperprolactinemia and it's symptoms.
Use While Breastfeeding:
The biggest reason why Cabergoline is admired by amateur and professional athletes is because it helps them reduce or eliminate the risks associated with excess prolactin that is common with use of harsh and aromatizable steroids like Trenbolone and Deca Durabolin.
Furthermore, this drug is also useful for treating sexual dysfunction caused by excess prolactin besides gaining an erection between orgasms and reducing recovery time after intense workouts or weight training and strength training exercises.
In addition to these advantages, the use of Dostinex is equally beneficial to combat estrogenic side effects such as oily skin, acne, gynecomastia, and bloating and treating health complications like galactorrhea and sexual dysfunction. It is also routinely indicated to patients with Parkinson's disease as it has the potential to work on information pathways and nervous system of the body.
Dostinex is also admired for its ability to make athletes feel 'full' that helps in minimizing food cravings without dieting discomfort.
Side Effects:
This medication is used to treat high levels of prolactin hormone in your body. High levels of prolactin in women can cause symptoms such as unwanted breast milk and missed periods and can cause difficulty becoming pregnant. High levels of prolactin in men can cause symptoms such as enlarged breasts and decreased sexual ability/desire. Cabergoline is an ergot medication and works by blocking the release of prolactin from the pituitary gland.
Some of the side effects that can occur with cabergoline may not need medical attention. As your body adjusts to the medicine during treatment these side effects may go away. Your health care professional may also be able to tell you about ways to reduce or prevent some of these side effects. If any of the following side effects continue, are bothersome or if you have any questions about them, check with your health care professional.
Lab Test Result:
Test Items |
Specification |
Results |
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Description |
White or almost white crystarlline powder |
Conforn |
||
Identify |
1. IR complies 2. X-Ray complies 3. HPLC complies |
Conforn Conforn Conforn |
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Water |
No more than 0.5% |
0.2% |
||
Reiated substances |
1.Allylamide (USP,rel,D) no more than 0.10% 2. Allyl DHLA(USP,rel,D) no more than 0.15% 3.Cabergoline oxide no more than 0.10% 4.Other impurities individually no more than 0.10% 5.Total no more than 0.50% |
0.02% Less than 0.02% Less than 0.02% Less than 0.02% 0.05% |
||
Assay(HPLC) |
98.0-102.0% |
99.5% |
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Opdical rotation |
-83-- -77 |
-78 |
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Residual Solvents |
1.Dichloromethane no more than 100ppm 2.Acetone no more than200ppm 3.Tert-butylmethylether no more than 200ppm 4.Xylene no more than 1500ppm 5.HEptane no more than 1000ppm |
Less than30ppm Less than20ppm Less than10ppm 110ppm Less than30ppm |
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Residue on ignition |
NO more than0.10 % |
0.02% |
||
Heavy metals |
NO more than 20ppm |
2ppm |
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Partcle size |
90%af particles no mone than 80μm |
Conform |
||
Bulk Density |
0.2~0.35g/em |
0.33g/em |
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Conclusion |
Conforn with USP38 Standard |
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Supervisor |
Yang Sun |
Analyst |
Sin Lee |
Anti-Estrogen Series |
|
Tamoxifen Citrate (Nolvadex) |
Dutasteride (Avodart) |
Clomifene Citrate (Clomid) |
Finasteride (Proscar) |
Letrozole (Femara) |
Formestane (Lentaron) |
Toremifene Citrate (Fareston) |
Cabergoline (Caber) |
Exemestane (Aromasin) |
Raloxifene Hydrochloride |
Anastrozole (Arimidex) |
Pramipexole |