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anti estrogen supplements,
anti estrogen products
Selective Estrogen Receptor Modulator (SERM) Toremifene Citrate / Fareston Powder
Toremifene Citrate is an oral selective estrogen receptor modulator (SERM) derived from
triphenylethylene. It is FDA approved for breast cancer treatment, and has possible medical uses
for prostate cancer. Bodybuilders will use this drug to combat gynecomastia (bitch tits), but it's
still very new to the scene and has some drawbacks.
It has already been covered that Toremifene is a SERM, and serves to block Estrogen at various
receptor sites in certain tissues within the body. As a layman explanation, Toremifene pretends to
be a 'fake' Estrogen that occupies Estrogen receptors within breast tissue. With these receptors
occupied by Toremifene, real Estrogen cannot perform their jobs there. Toremifene does not
reduce total blood plasma levels of Estrogen. In addition to being antagonistic to Estrogen
receptors in breast tissue, it is also antagonistic to Estrogen at the hypothalamus gland this
essentially 'tricks' the hypothalamus into thinking there is little or no circulating Estrogen levels in
the body, causing it to increase its manufacture of Testosterone so that it can utilize aromatization
to restore these levels.
Toremifene is also agonistic to Estrogen receptors in other tissues in the body. This means that
whileToremifene will act as an anti-estrogen in breast tissue and the hypothalamus, it will act as
an Estrogen within the liver. This can have beneficial impacts especially during an anabolic
steroid cycle, such as improving and shifting cholesterol levels into a more favorable range.
In the fight against breast cancer, standard Fareston doses will normally be 60mg per day. The
total duration of use is unpredictable and will be based on patient need. It's not uncommon for
treatment to last a year or two and then AI's to be added if needed. Once the cancer is in
remission, compounds like Fareston are commonly used to support the improved state.
For the anabolic steroid user combating gynecomastia, standard Fareston doses will fall in the
30-60mg per day range and will work very well for most men. If this is not enough protection, while
you could try increasing the dose your best bet would be to move to AI use. You will find Fareston
works very well in combating gynecomastia due to the use of any testosterone, Dianabol and
Anadrol. You will also find it works well with Equipoise and Deca Durabolin. However, as Deca
Durabolin is also a progestin, men who are very sensitive to that hormone may need an AI. The
same can be said of the Trenbolone hormone. Trenbolone does not aromatize, but it is a
progestin. Further, the use of an aromatizing steroid with a compound like Trenbolone can
increase the risk of gynecomastia in some men. While many will not need gynecomastia
protection due to progestins and will get by with SERM's to combat aromatase, some sensitive
men will need an AI. Regardless, if Fareston works for you it will cover the entire breadth of the
cycle from start to finish.
For bodybuilding purposes, a dose of 40-60 mg/day seems to be a good starting point. If the
user is trying to fight existing gynecomastia, they may choose to double the dose and add an
aromatase inhibitor like Aromasin with it. For PCT, some users will kick-start with 100-120
mg/day and then lower to 40-60 mg/day for 4-6 weeks.
Tamoxifen Citrate (Nolvadex)
Clomifene Citrate (Clomid)
Toremifene Citrate (Fareston)
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